Alkynyl Benzoxazines and Dihydroquinazolines as Cysteine Targeting Covalent Warheads and Their Application in Identification of Selective Irreversible Kinase Inhibitors

Journal of the American Chemical Society

Kirsten McAulay, Emily A Hoyt, Morgan Thomas, …, Richard A Ward, Michael J Waring, Jason G Kettle

• DOI: 10.1021/jacs.9b13391
• PMID: 32412754